Magnesium stearate safety, side
effects, toxicity, problems and review of studies
Is magnesium stearate found in supplement capsules safe?
Are there web sites that are spreading false safety concerns about this ingredient?
December 6 2017 by
Ray Sahelian, M.D.
Stearic acid is a common fatty acid found in significant amounts in meat, poultry, fish, eggs, butter, grains, and milk products. Some websites have misleading information regarding the safety of magnesium stearate. Some of these sites claim magnesium stearate, even in as small an amount as a few milligrams. as found in dietary supplement capsules, is dangerous.
There is no evidence this is true, particularly the tiny amounts found in supplements. I am not aware of any human studies that show MS, in the small amounts found in capsules, has any side effects or causes any harm.
There is no evidence that
small amounts of stearic acid are harmful. If anyone knows of a human study that
indicates magnesium stearate, in the small amounts found in capsules, when taken
orally in supplement form, has shown
to have harmful effects, email me. I have searched extensively and not seen any such
clinical trials. I believe there is misinformation on web sites that claim this
substance is harmful.
Much of this mis-information
is posted by companies who are trying to differentiate themselves from other
vitamin companies by providing products that are free of mag stearate, perhaps
because they are not able to compete solely on the actual effectiveness of their
products. If anyone tells you
magnesium stearate in the extremely small amounts found in capsules is harmful, challenge
them to provide you with a human study that proves their point -- they will not
be able to.
For some consumers this whole issue has become almost a psychological obsession
going way beyond any logical reasoning. Some people regularly eat a piece of
pie, cookie, or other sweet or junk food, or consume chocolate (which has tons
of stearic acid) without any concerns, but get all worked up about insignificant
amounts found in capsules. It defies logic.
Most dietary supplement capsules have about 500 mg of herbs or
nutrients and perhaps 10 mg or less of magnesium stearate. Since magnesium
mineral is part of the overall weight of the molecule, the amount of
stearate alone is even less than 10 mg. One kilogram equals 1000 grams, and one gram equals 1000 mg. A few milligrams is an insignificant amount compared to the millions of
milligrams of food we consume a day.
I have been taking dietary supplements for more than thirty years
and I know older patients who have been taking a handful of vitamin capsules with
magnesium stearate every day for more than 40 or 50 years and they are in their
80s and 90s (even a few who are over a 100 years old) and
in good health. If MS was so toxic as some claim, how come none of these vitamin users have
become ill after consuming these ms-containing capsules daily for several
decades?
I question the medical
acumen of any nutritionist or doctor who claims this substance poses a danger in
the miniscule amounts found in vitamin / supplement pills.
What is it?
Magnesium stearate is a white substance that has two
equivalents of stearate and one magnesium cation. It is safe for human
consumption. It is often used as a filling agent
in the manufacture of supplement capsules. This substance has lubricating properties and prevents ingredients from sticking to
manufacturing equipment during the compression of chemical powders into capsules
or tablets. Most pharmaceutical formulations include a certain amount of
lubricant to improve their flowability and prevent their adhesion to the
surfaces of processing equipment.
Chocolate contains cocoa butter, which is high in saturated fat.
About a third of the fat in chocolate is in the form of stearic acid.
Stearic acid in food
Stearic acid is the most common of the long-chained fatty acids. It is
found in many foods including vegetable and animal oils, beef fat, and cocoa
butter. A person who eats a chocolate bar will ingest hundreds of times more stearic acid than someone taking a dietary supplement with magnesium stearate.
Safety of magnesium stearate and
stearic acid, risk or danger, side effects and toxicity?
I am not aware of any human studies that show MS, in the small amounts found in capsules, has any side effects,
poses risks, danger, safety issues
or causes any bodily harm. There is no evidence that small amounts of stearic acid are
harmful. The studies below prove that stearic acid, even in moderate amounts,
has not been shown to be harmful.
A stearic acid-rich diet improves thrombogenic and
atherogenic risk factor profiles in healthy males.
Eur J Clin Nutrition. 2001.
To determine whether healthy males who consumed increased amounts of dietary
stearic acid compared with increased dietary palmitic acid exhibited any changes
in their platelet aggregability, platelet fatty acid profiles, platelet
morphology, or haemostatic factors. Results from this study indicate that
stearic acid (19g/day) in the diet has beneficial effects on thrombogenic and
atherogenic risk factors in males. The food industry might wish to consider the
enrichment of foods with stearic acid in place of palmitic acid and trans fatty
acids.
Influence of stearic acid on hemostatic risk factors in
humans.
Lipids. 2005. The Research Department of Human
Nutrition, Centre of Advanced Food Research, The Royal Veterinary and
Agricultural University, Frederiksberg, Denmark.
Here I report the results of three controlled,
human dietary intervention studies, which used a randomized crossover design to
investigate the hemostatic effects of stearic acid-rich test diets in healthy
young men. A diet high in stearic acid (shea butter) resulted in a 13% lower
fasting plasma FVIIc than a high palmitic acid diet, and was 18% lower than a
diet high in myristic and lauric acids after 3 wk of intervention. The present
investigations did not find dietary stearic acid to be more thrombogenic, in
either fasting effects compared with other long-chain fatty acids, or in acute
effects compared with dietary unsaturated FA, including trans monounsaturated
FA.
Q. I recently read that Magnesium Stearate is made from
cottonseed oil with pesticides and that it is toxic to the liver. Is this true?
A. It is not toxic to the liver.
Statement by chemical manufacturer Hummel Croton Inc.,
South Plainfield, NJ
Hazards Identification regarding magnesium stearate:
Acute health effects: Irritating to the skin and eyes on contact. Inhalation
will cause irritation to the lungs and mucus membrane. Irritation to the eyes
will cause watering and redness. Reddening, scaling, and itching are
characteristics of skin inflammation. Follow safe industrial hygiene practices
and always wear protective equipment when handling this compound.
Chronic health effects: This product has no known chronic effects. Repeated or
prolong exposure to this compound is not known to aggravate medical conditions.
Acute health effects: This product is not listed by NTP, IARC or regulated as a
carcinogen by OSHA.
Absorption issues
Some consumers having read on websites that have unreliable information that MS
hinders absorption of the active ingredients. This is not true. People take
their supplements with food (chicken, chocolate) that contains hundreds of times
the stearic acid found in supplements, yet absorb the herbs or vitamins quite
well. I have seen no evidence that the intake of the tiny amounts of mag stearate in capsules interferes with intestinal absorption of nutrients.
Anyone who makes this claim needs to show scientific proof with several studies done in
humans. Anyone who makes this claim does not have an understanding regarding
human intestinal absorption. The intestines are very long and contain an
enormous area of absorptive space whereas the amount of MS is so minimal it
would hardly take up any space in the vast intestinal area of absorptive
ability.
Allergy
There have been rare reports of magnesium stearate allergy.
J Biological Regul Homeost Agents. 2012. Magnesium stearate: an underestimated allergen. Magnesium stearate is a substance often used as a diluent in the manufacture of medical tablets, capsules and powders. Moreover it is usually found as a food additive or pharmaceutical excipient. We report the first case of a 28 years old woman affected by an allergic reaction from this substance with an urticarial manifestation.
Emails
Q. Thank you for your Passion Rx. It actually
works! Here is a quote from a website, "The Truth About Vitamin
Supplements: Check your vitamin labels. Do they contain Magnesium Stearate or
Stearic Acid? Studies by the University of Texas Health Science Center and the
East Carolina University School of Medicine reveal that these toxic excipients
cause a rapid collapse of T-cell membrane function and cell death; therefore
suppressing the immune system. (Immunology, 1990, July). It is estimated that
90% of the vitamin and mineral products consumed today contain stearates.
These are used as binders in tablets and in the processing of gelatin
capsules. Consumers often take handfuls of capsules and tablets to get vitamins,
minerals and other key nutrients from supplements that contain stearates, and
instead, in reality, get a powerful immune suppressive treatment. For more
information on this topic and copies of the above-quoted studies as well as
other studies and warnings concerning stearates, send an email to Quantum
Nutrition Labs' nutritional supplements. Our products are 100% free of toxic
excipients, including magnesium stearate or stearic acid."
A. Much of the misinformation about the safety or toxicity is
posted by companies who are trying to make themselves different from other
vitamin companies by providing products that are free of this ingredient. The study
referred to by this company was actually done in a cell culture. Below is the study that is referred to and my comments.
Molecular basis for the immunosuppressive action of stearic acid on T cells.
Immunology. 1990. Department of Microbiology and
Immunology, East Carolina University School of Medicine, Greenville.
Studies were performed to determine the mechanism by which stearic acid
(18:0) selectively inhibits T-dependent immune responses in vitro. Incubation of
mitogen-activated B and T cells with stearic acid resulted in dissimilar
patterns of incorporation of the saturated fatty acid into their membranes.
High-performance liquid chromatography (HPLC) analyses of T cells showed an
accumulation of disaturated 18:0-containing phosphatidylcholine (PC) that
replaced normal cellular PC. Less significant quantities of the same PC species
were seen to accumulate in B-cell membranes; rather, they increased their
proportion of oleic acid containing PC. The different lipid compositions
of the lymphocyte cell membranes after exposure to 18:0 were correlated with
their plasma membrane potentials. In T cells, the accumulation of disaturated,
18:0-containing PC coincided with a rapid (within 8 hr) collapse of membrane
integrity, as determined by flow cytometry. The collapse of membrane integrity
was found to be time and dose dependent. No such depolarization was observed in
B cells which, by virtue of their desaturating ability, were able to avoid
incorporating large amounts of disaturated 18:0-containing phospholipids into
their membranes. It is proposed that a lack of stearoyl-CoA desaturase in T
cells precludes them from desaturating exogenously derived 18:0, thus leading to
increased proportions of 18:0-containing disaturated PC in their cell membranes.
The increased abundance of this PC species may enhance membrane rigidity to an
extent that plasma membrane integrity is significantly impaired, leading to a
loss of membrane potential and ultimately cell function and viability.
Comments: This study is totally irrelevant to what would occur in the human body from the tiny amounts of stearic acid ingested in capsules. If you directly put a particular nutrient, vitamin, fatty acid, amino acid, medication, herb or any substance in a high enough dosage directly in a cell culture you will get results that have nothing to do with what happens when a tiny amount is ingested as part of a medicine, supplement, or through diet and is diluted and distributed to trillions of cells. For instance, you can kill a cell if you put too high an amount of fish oil fatty acids near it in a cell culture, but that does not mean fish oil fatty acids, the omeag-3s, are harmful to you when ingested in reasonable amounts - in fact omega-3s are healthy fatty acids. People or companies who use this type of in vitro study to make such a leap either do not understand medicine or science, or are purposely misleading consumers for marketing reasons.
Q. Are these studies not valid?
“Stearic Acid inhibits T-cell dependent immune responses. Plasma membrane
integrity is significantly impaired, leading to a loss of membrane potential and
ultimately cell function and viability.” Tebbey PW, Buttke TM, “Molecular Basis For The Immunosuppressive Action of
Stearic Acid on T cells” (Immunology, 1990 July. When cells were exposed to stearic acids and palmitic
acids, there was a dramatic loss of cell viability after 24 hours.”
Ulloth, JE, Casiano CA, De Leon M. Department of
Microbiology and Immunology, East Carolina University School of Medicine.
“T-helper cells become the target of stearic acid.”
“The addition of palmitate or stearate to cultured cells led to activation of a
death program with a morphology resembling that of apoptosis. Palmitates and
stearates caused cardiac and other types of cells to undergo programmed cell
death.”
Sparagna, GC, Hickson-Bick, DL, Department of Pathology and Medicine, University
of Texas Health Science Center, Houston. American Journal of Medical Science,
1999.
A. You can put an excess of
any healthy substance, including fish oils, around cells in a Petri dish and the
cells can die. This does not mean that fish oils are harmful when ingested in
reasonable amounts. What happens in an isolated cell in a Petri dish has little relevance to the actual ingestion of that substance since the
dilution of the substance that ends up in trillions of cells in the body makes
it insignificant.
Q. Can you comment on these I found on some website?
“Stearic Acid, Magnesium Stearate, Calcium Stearate, Palmitate, and Hydrogenated
Vegetable Oils are lubricants which enable manufacturing equipment to run more
efficiently but inhibit eventual dissolution of the nutrient. Stearic acid may
prevent absorption by individuals with compromised digestive systems. Magnesium
stearate and stearic acid also present the problem that delivery of the active
ingredient may be considerably further down the intestinal tract than the site
originally intended. This may result in the nutrient being delivered away from
its optimal absorption site. Not only can this impede absorption, in some cases
it might be harmful to the liver.”
Czap, AL. Townsend Letter For Doctors and Patients, 1999.
Consumers often take handfuls of capsules to get nutrients from supplements
containing magnesium stearate or stearic acid and instead, get a powerful immuno
suppressive treatment!
A. The statements above are probably written by someone who
does not have a good understanding of the human body, physiology, metabolism and
digestion.
Q. I recently bought a hoodia
product. I was disappointed to see magnesium stearate (from
vegetable products ) on the label. Rival products claim hoodia
containing magnesium stearate as POISON ! I subsequently did some research on
various sites and was relieved to find out it was harmless
in the manufacture of supplement tablets.
Q. Most of the
time magnesium stearate is made by subjecting cottonseed or palm oil to high
heat and pressure in the presence of a metal (in this case magnesium) catalyst
for several hours. This creates a hydrogenated saturated fat. I did the math and
it follows that if each 1000mg capsule has approximately 2% magnesium stearate
in it ( this seems to be about average) that means 20 mg of the capsule is
hydrogenated fat. If I take ten capsules a day I would be ingesting about
73,000mg of hydrogenated fat per year or about 2.5 ounces. Like most people who pay
attention to their health and take supplements, I take a lot more than ten
capsules a day. As a person who reads labels at the grocery store and promptly
rejects any foodstuff with hydrogenated oil in it, why would I take a supplement
with hydrogenated oil in it?
A. The amount of stearate consumption is even less since magnesium
is part of the weight. Therefore, even if there is 20 mg or so of MS in a 1,000 mg supplement capsule,
some of that weight is a healthy mineral. Some people get quite obsessed
about minutia that, practically speaking, have little or no influence on their
health. One could get worried about these tiny amounts that is not likely to have any health effects yet have no
concerns about getting in the car to drive to the local movie theatre. The risk
of a car accident with bodily harm or inhaling pollutants while on the road are
much more likely to occur than the minute amounts of magnesium stearate causing
harm to health. If a person is that worried about every possible harm that could
occur to them, then they would stay home and not even go out of the house. Then
again that has its own risks since one could become vitamin D deficient due to
lack of sunlight and possibly get depressed due to lack of human interaction. The amount of hydrogenated oils
you mention as a result of ingesting 10 capsules a day about the same or less
than eating half a donut over a period of one year. (See an email below that
questions the presence of hydrogenated oils in mag stearate.) If your diet is so
perfect (with absolutely no sugar, bad fats, cookies, cakes, ice cream, etc)
that eating the equivalent of half a donut over a period of year would concern
you, then you may look to find supplements that do not contain it. How many
people can truly claim that throughout the whole year they do not ingest any ice
cream, regular soda, cookies, pastries, a piece or birthday cake, white bread,
chocolate, more than a cup of coffee a day, cream added to the coffee,
artificial sweeteners, margarine, or any type of unhealthy food? I think
drinking several ounces of fruit juice at one time is a much more significant
health issue since it raises blood sugar levels and promotes an excess insulin
response. If a person is
taking more than 10 capsules of supplements a day, there is a significantly
higher risk of side effects from the active ingredients in all of these pills
rather than the insignificant amount of fillers or lubricants. It often surprises me how some people go to great lengths trying to avoid ingesting something that has practically no harm yet do
not realize there is a higher risk of harm from so many other activities they do
routinely, for instance driving for leisure or even going skiing.
Q. I work for a vitamin company and have been doing a little
reading up on these substances. Stearic acid / mag stearate does not have any trans fatty acids in it. The
person asking the question is making it sound as if there is a concern about
this, and your response implies that there is so little, that it should not be a
concern. It’s my understanding, that there is 0 trans fatty acids. The trans
fatty acids are formed when the oil is only partially hydrogenated. This
Statement by Now Foods talks about it a little and says there are 0 trans fats.
http://www.nowfoods.com/Quality/QualityNotes/M093528.htm
Perhaps you could change that response? This seems to be coming
more of an issue.
A. Yes, you are right, I am assuming that there are are some
hydrogenated oils in the magnesium stearate since high temperatures may be used
in the preparation. I would still like to see an independent analysis to
determine whether any of the stearic acid is hydrogenated. Not that it matters
much since the amounts that are consumed are so tiny to be practically
irrelevant.
Q. My Grandmother became
worried when an associate told her she was killing herself because she took 30
to 60 capsules a day of MSM (Organic Sulfur) which contained magnesium stearate
in each capsule. My grandmother swears by this stuff; she's been taking it for
years and her skin is flawless. She's 75 and looks 45. She's very active and
doesn't have joint pain like most of her friends. If she's taking 30 to 60 capsules a day of MSM
with MS in the capsules, is this toxic in your opinion?
A. She has been taking all these capsules for all these years and yet, as
you mention, she is vibrant and 75 years old. If it were toxic she would have
had some negative symptoms or side effects by now.
Q. 2012 - Dr. Mercola sent out an email
warning against using supplements that use magnesium stearate or stearic acid as
filler. There are other sources besides Dr. Mercola that
also warn of toxicity. Here is information taken
from his website, "Steer Clear of
Magnesium Stearate, I realize that there is very little research published on
this. The bottom line is actually quick and simple. Some highly respected
clinicians like Dr. Klinghardt and others have extensive experience with this
issue."
A. As with many topics, health, politics, religion, etc, there
are different viewpoints held by different people. It is up to each individual
to learn as much as they can and then come to their
own conclusion on whose opinion they trust. I have personally taken supplements
with magnesium stearate for more than 30 years without any ill effects.
Q. Email received 2015: Please let me know your
response to Dr. Mercola’s statements on the safety of magnesium stearate. He
claims that magnesium stearate causes damage to T cells and has other harmful
effects on the human body.
A. As of 2017, I stand by my views as written on this page.
Q. I am the Vice-President of R&D for a vitamin
corporation. We are a large Private Label manufacturer in the US and have been
seeing an increase in customer requests for the substitution of magnesium
stearate and stearic acid in formulations. As you know, the formulation benefits
of both are important and necessary to a cost-effective product and attempting
to substitute with an inferior “natural” substitute (ie. Rice Hulls) is
problematic in production and not a cost effective solution. I have read your
post which is very informative and useful in the defense of its use in dietary
supplements. I see that as of 2017, you are still standing my your statements
within the article. I am attempting to create a logical defense of its position
for our customers and would like to ask your permission if I could reference
your article in my conversation.
A. Yes, please feel free to reference my article. I will update as
I come across more information.